EP4 receptor antagonist 4
Modify Date: 2024-09-18 08:19:05
EP4 receptor antagonist 4 structure
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Common Name | EP4 receptor antagonist 4 | ||
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| CAS Number | 691869-12-2 | Molecular Weight | 318.39 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C19H14N2OS | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of EP4 receptor antagonist 4EP4 receptor antagonist 4 is an EP4 receptor agonist with the human pEC50 value of 6.3[1]. |
| Name | EP4 receptor antagonist 4 |
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| Description | EP4 receptor antagonist 4 is an EP4 receptor agonist with the human pEC50 value of 6.3[1]. |
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| Related Catalog | |
| Target |
EP4:6.3 (pEC50) |
| In Vitro | EP4 receptor antagonist 4 (24 h) treatment shows agonism in HEK293 cells stably transfected with hEP4[1]. EP4 receptor antagonist 4 (30 min) treatment shows agonism (pEC50<5) and antagonism (pIC50<5)[1]. Cell Viability Assay[1] Cell Line: HEK293 cells Concentration: Incubation Time: 24 hours Result: Exhibited the human pEC50 value of 6.3. |
| References |
[1]. Joannes Theodorus Maria Linders, et al. Bicyclic derivatives as ep4 agonists. WO2008092860A1 |
| Molecular Formula | C19H14N2OS |
|---|---|
| Molecular Weight | 318.39 |