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Abarelix acetate

Abarelix acetate用途

Abarelix acetate is a synthetic third generation gonadotropin-releasing hormone receptor (GnRHR) antagonist. It increases histamine release from rat peritoneal mast cells in vitro and from a human skin model ex vivo. In vivo, abarelix decreases plasma luteinizing hormone (LH) levels six hours post-treatment in castrated rats, with levels returning to baseline within 24 hours.3 Abarelix (2 mg/kg) also transiently decreases plasma testosterone levels in intact rats, with levels returning to baseline within seven days post-treatment. Formulations containing abarelix have previously been used in the treatment of advanced prostate cancer.

Abarelix acetate名称

[ CAS 号 ]:
785804-17-3

[ 英文名 ]:
Abarelix acetate

[英文别名 ]:

Abarelix acetate物理化学性质

[ 分子式 ]:
C74H99ClN14O16

[ 分子量 ]:
1476.115

[ 精确质量 ]:
1474.705200

推荐生产厂家/供应商:

公司名:上海化源世纪贸易有限公司

区域:上海市普陀区

价格:

联系人:徐乾明

产品详情:Abarelix (acetate)


公司名:上海脉铂医药科技有限公司

区域:上海市嘉定区

价格:
¥1540.0/1mg ¥13860.0/25mg ¥6930.0/10mg ¥需询单/10mg

联系人:李先生

产品详情:Abarelix (acetate)


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Abarelix acetate供应商


相关化合物

[Abarelix acetate]化源网提供Abarelix acetateCAS号785804-17-3,Abarelix acetateMSDS及其说明、性质、英文名、生产厂家、作用/用途、分子量、密度、沸点、熔点、结构式等。CAS号查询Abarelix acetate上化源网,专业又轻松。>>电脑版:Abarelix acetate

标题:785804-17-3_Abarelix acetateCAS号:785804-17-3_Abarelix acetate【结构式 性质 英文】 - 化源网 地址:https://www.chemsrc.com/amp/cas/785804-17-3_1567689.html