149669-43-2

• 常用中文名：5-氟-3-(4-哌啶)-吲哚
• 常用英文名：5-Fluoro-3-(piperidin-4-yl)-1H-indole
• CAS号：149669-43-2
• 分子式：C₁₃H₁₅FN₂
• 分子量：218.27000
• 发布时间：2018-07-20 17:09:56
• 更新时间：2024-01-10 10:15:12

名称

• 中文名: 5-氟-3-(4-哌啶)-吲哚
• 英文名: 5-Fluoro-3-(piperidin-4-yl)-1H-indole
• 中文别名: 5-氟-3-(哌啶-4-基)-1H-吲哚
• 英文别名: 5-fluoro-3-piperidin-4-yl-1H-indole

物化性质

• 分子式: C₁₃H₁₅FN₂
• 分子量: 218.27000
• 精确质量: 218.12200
• PSA: 27.82000
• LogP: 3.10280
• 储存条件: 室温，避光，保存于惰性气体中

合成路线

127626-06-6 ~% 149669-43-2

文献：Eli Lilly and Company Patent: US5708187 A1, 1998 ; US 5708187 A Title/Abstract Full Text Show Details Eli Lilly and Company Patent: US5708008 A1, 1998 ; US 5708008 A

194036-50-5 ~% 149669-43-2

文献：JANSSEN PHARMACEUTICA, N.V. Patent: WO2007/50381 A2, 2007 ; Location in patent: Page/Page column 37-38 ; WO 2007/050381 A2

399-52-0 ~% 149669-43-2

文献：Wrobel, Martyna Z.; Chodkowski, Andrzej; Herold, Franciszek; Gomolka, Anna; Kleps, Jerzy; Mazurek, Aleksander P.; Plucinski, Franciszek; Mazurek, Andrzej; Nowak, Gabriel; Siwek, Agata; Stachowicz, Katarzyna; Slawinska, Anna; Wolak, Malgorzata; Szewczyk, Bernadeta; Satala, Grzegorz; Bojarski, Andrzej J.; Turlo, Jadwiga European Journal of Medicinal Chemistry, 2013 , vol. 63, p. 484 - 500

399-52-0 40064-34-4 ~67% 149669-43-2

文献：Pages Santacana, Lluis; Fonquerna Pou, Silvia; Puig Duran, Carles; Fernandez Forner, Dolors Patent: US2002/147344 A1, 2002 ;

41979-39-9 ~% 149669-43-2

文献：Fonquerna, Silvia; Miralpeix, Montse; Pages, Lluis; Puig, Carles; Cardus, Arantxa; Anton, Francisca; Cardenas, Alvaro; Vilella, Dolors; Aparici, Monica; Calaf, Elena; Prieto, Jose; Gras, Jordi; Huerta, Josep M.; Warrellow, Graham; Beleta, Jorge; Ryder, Hamish Journal of Medicinal Chemistry, 2004 , vol. 47, # 25 p. 6326 - 6337

41661-47-6 ~% 149669-43-2

文献：Wrobel, Martyna Z.; Chodkowski, Andrzej; Herold, Franciszek; Gomolka, Anna; Kleps, Jerzy; Mazurek, Aleksander P.; Plucinski, Franciszek; Mazurek, Andrzej; Nowak, Gabriel; Siwek, Agata; Stachowicz, Katarzyna; Slawinska, Anna; Wolak, Malgorzata; Szewczyk, Bernadeta; Satala, Grzegorz; Bojarski, Andrzej J.; Turlo, Jadwiga European Journal of Medicinal Chemistry, 2013 , vol. 63, p. 484 - 500

上下游产品

上游产品  5
127626-06-6 399-52-0 40064-34-4 41979-39-9
41661-47-6
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