Mutation Research/Fundamental and Molecular Mechanisms of Mutagenesis 1991-12-01

Mutagenicity of 2-methylacrolein, 2-ethylacrolein and 2-propylacrolein in Salmonella typhimurium TA100. A comparative study.

T Neudecker, E Eder, C Deininger, D Henschler

Index: Mutat. Res. 264(4) , 193-6, (1991)

Full Text: HTML

Abstract

The C2-alkylated acrolein derivatives 2-methylacrolein, 2-ethylacrolein and 2-propylacrolein are mutagenic in Salmonella typhimurium TA100. They are direct mutagens, their mutagenic potency being inversely proportional to the size of the alkylating substituent in the C2 position. In the presence of S9 mix, the mutagenicity of all these substances is considerably reduced; the reduction in mutagenicity is inversely proportional to the direct mutagenic potential of the substance. As shown for 2-methylacrolein, the reduction in mutagenicity is dependent on the concentration of S9 in the S9 mix and is not significantly influenced by heat inactivation of the S9 mix or by addition of TCPO, an inhibitor of epoxide hydrolase, to the testing system. There are no indications of enzymatic activation by the metabolizing microsomal system.


Related Compounds

Related Articles:

An efficient approach to Aspidosperma alkaloids via [4 + 2] cycloadditions of aminosiloxydienes: stereocontrolled total synthesis of (+/-)-tabersonine. Gram-scale catalytic asymmetric syntheses of (+)-tabersonine and (+)-16-methoxytabersonine. Asymmetric syntheses of (+)-aspidospermidine and (-)-quebrachamine.

2002-05-01

[J. Am. Chem. Soc. 124(17) , 4628-41, (2002)]

Immunological response from an entirely carbohydrate antigen: design of synthetic vaccines based on Tn-PS A1 conjugates.

2009-07-22

[J. Am. Chem. Soc. 131(28) , 9622-3, (2009)]

Mutagenicity of 2-alkylpropenals in Salmonella typhimurium strain TA 100: structural influences.

2001-01-01

[Environ. Mol. Mutagen. 37(4) , 324-8, (2001)]

Repeated exposure to alpha-ethylacrolein vapour: subacute toxicity study in rats.

1981-01-01

[Toxicology 22(1) , 79-87, (1981)]

More Articles...