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KDM4-IN-3

Names

[ CAS No. ]:
1068515-53-6

[ Name ]:
KDM4-IN-3

Biological Activity

[Description]:

KDM4-IN-3 is a KDM4 inhibitor that exhibits improved potency in biochemical assays, is cell-permeable, and kills prostate cancer cells at low micromolar concentrations.

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Histone Demethylase

[References]

[1]. Carter DM, et al. Enhanced Properties of a Benzimidazole Benzylpyrazole Lysine Demethylase Inhibitor: Mechanism-of-Action, Binding Site Analysis, and Activity in Cellular Models of Prostate Cancer. J Med Chem. 2021 Oct 14;64(19):14266-14282.

Chemical & Physical Properties

[ Molecular Formula ]:
C17H14N4O

[ Molecular Weight ]:
290.32

Related Compounds