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Lys-[Hyp3]-Bradykinin

Names

[ CAS No. ]:
113662-39-8

[ Name ]:
Lys-[Hyp3]-Bradykinin

Biological Activity

[Description]:

Lys-[Hyp3]-Bradykinin a Bradykinin (HY-P0206) agonist. Lys-[Hyp3]-Bradykinin is a kinin, it can be isolated from human urine. Lys-[Hyp3]-Bradykinin can be used for the research of inflammation[1].

[Related Catalog]:

Research Areas >> Inflammation/Immunology
Signaling Pathways >> GPCR/G Protein >> Bradykinin Receptor

[In Vitro]

Lys-[Hyp3]-Bradykinin (0.1 nM-1 μM) displaces [3H]-BK from solubilized binding sites of cultured human fibroblasts with a dose-dependent maner[1]. Lys-[Hyp3]-Bradykinin (0.5 μM; 7 min) increases CAMP level up to an 16-fold in human fibroblasts[1].

Chemical & Physical Properties

No Any Chemical & Physical Properties


Related Compounds