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Pregabalin arenacarbil

Names

[ CAS No. ]:
1174748-30-1

[ Name ]:
Pregabalin arenacarbil

[Synonym ]:
(3S)-3-[({[(1R)-1-(Isobutyryloxy)ethoxy]carbonyl}amino)methyl]-5-methylhexanoic acid
Hexanoic acid, 5-methyl-3-[[[[(1R)-1-(2-methyl-1-oxopropoxy)ethoxy]carbonyl]amino]methyl]-, (3S)-

Biological Activity

[Description]:

Pregabalin arenacarbil is a prodrug of Pregabalin.Pregabalin is an analog of gamma-aminobutyric acid (GABA) for the research of post herpetic neuralgia, peripheral diabetic neuropathy,fibromyalgia and epilepsy[1].

[Related Catalog]:

Signaling Pathways >> Membrane Transporter/Ion Channel >> GABA Receptor
Research Areas >> Metabolic Disease
Signaling Pathways >> Neuronal Signaling >> GABA Receptor

[References]

[1]. Gallop, Mark A, et al.Method for the enzymatic kinetic resolution of acyloxyalkyl thiocarbonates used for the synthesis of acyloxyalkyl carbamates.WO2009094569A2

Chemical & Physical Properties

[ Density]:
1.1±0.1 g/cm3

[ Boiling Point ]:
457.5±30.0 °C at 760 mmHg

[ Molecular Formula ]:
C15H27NO6

[ Molecular Weight ]:
317.38

[ Flash Point ]:
230.5±24.6 °C

[ Exact Mass ]:
317.183838

[ LogP ]:
2.99

[ Vapour Pressure ]:
0.0±2.4 mmHg at 25°C

[ Index of Refraction ]:
1.468

Related Compounds