TRPV antagonist 1

Names

[ CAS No. ]:
1192871-27-4

[ Name ]:
TRPV antagonist 1

Biological Activity

[Description]:

TRPV antagonist 1 is a transient receptor potential vanilloid (TRPV) antagonist, with an IC50 of < 250 nM.

[Related Catalog]:

Signaling Pathways >> Membrane Transporter/Ion Channel >> TRP Channel

Research Areas >> Others

[Target]

IC50: < 250 nM (TRPV)[1]

[References]

[1]. Reilly RM, et al. Analgesic potential of TRPV3 antagonists. Curr Top Med Chem. 2011;11(17):2210-5.

[Related Small Molecules]

capsaicin | Capsazepine | EIPA | Diphenyleneiodonium chloride | HC-030031 | SKF-96365 | HC 067047 | AMG 9810 | GSK-1016790A | SAR7334 | PF-4840154 | RN-1734 | AMG-517 | SB-366791 | IcilinAG-3-5

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₆H₂₁F₃N₂O₄S

[ Molecular Weight ]:
514.52

TRPV antagonist 1

Names

Biological Activity

Chemical & Physical Properties

Related Compounds