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GCPII-IN-1 TFA

Names

[ CAS No. ]:
1269794-89-9

[ Name ]:
GCPII-IN-1 TFA

Biological Activity

[Description]:

GCPII-IN-1 TFA is a glutamate carboxypeptidase II (GCPII, or PSMA) inhibitor scaffold with a Ki of 44.3 nM[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Metabolic Enzyme/Protease >> Carboxypeptidase

[References]

[1]. Jan Tykvart, et al. Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. Bioorg Med Chem. 2014 Aug 1;22(15):4099-108.

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₄H₂₂F₃N₃O₉

[ Molecular Weight ]:
433.33

Related Compounds