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Endomorphin 2 TFA

Names

[ CAS No. ]:
1276124-00-5

[ Name ]:
Endomorphin 2 TFA

Biological Activity

[Description]:

Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Opioid Receptor
Signaling Pathways >> Neuronal Signaling >> Opioid Receptor
Research Areas >> Neurological Disease

[Target]

Ki: 20-30 nM (kappa3 opioid receptor)[1]


[References]

[1]. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.

Chemical & Physical Properties

[ Molecular Formula ]:
C34H38F3N5O7

[ Molecular Weight ]:
685.69

[ Storage condition ]:
2-8℃

Related Compounds