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5-HT2A receptor agonist-3

Names

[ CAS No. ]:
1391499-52-7

[ Name ]:
5-HT2A receptor agonist-3

Biological Activity

[Description]:

5-HT2A receptor agonist-3 is the most selective agonist for the human 5-HT2A receptor yet discovered, with a Ki of 2.5 nM, and with 124-fold selectivity for 5-HT2A over the structurally similar 5-HT2C receptor[1].

[Related Catalog]:

Research Areas >> Others
Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor
Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor

[Target]

2.5 nM (human 5-HT2A)


[References]

[1]. Juncosa JI Jr, et al. Extensive rigid analogue design maps the binding conformation of potent N-benzylphenethylamine 5-HT2A serotonin receptor agonist ligands. ACS Chem Neurosci. 2013;4(1):96-109.  

Chemical & Physical Properties

[ Molecular Formula ]:
C21H26BrNO3

[ Molecular Weight ]:
420.34

Related Compounds