Tasipimidine sulfate

Names

[ Name ]:
Tasipimidine sulfate

Biological Activity

[Description]:

Tasipimidine sulfate is an orally active and selective α2A-adrenoceptor agonist with a pEC50 of 7.57 against human α2A-adrenoceptor. Tasipimidine sulfate can be used for situational anxiety and fear research[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Adrenergic Receptor

Research Areas >> Neurological Disease

[Target]

human α2A-adrenoceptor:7.57 (pEC50)

rodent α2D-adrenoceptor:6.56 (pEC50)

human α2C-adrenoceptor:6.29 (pEC50)

human α2B-adrenoceptor:6.00 (pEC50)

[References]

[1]. Lehtimäki J, et al. Tasipimidine-the pharmacological profile of a novel orally active selective α2A-adrenoceptor agonist. Eur J Pharmacol. 2022 May 15;923:174949.

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₃H₁₈N₂O₆S

[ Molecular Weight ]:
330.36

Tasipimidine sulfate

Names

Biological Activity

Chemical & Physical Properties

Related Compounds