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BET-BAY 002

Names

[ CAS No. ]:
1588521-78-1

[ Name ]:
BET-BAY 002

[Synonym ]:
(4R)-6-(4-Chlorophenyl)-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4H-[1,2,4]triazolo[4,3-a][1]benzazepine
4H-[1,2,4]Triazolo[4,3-a][1]benzazepine, 6-(4-chlorophenyl)-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-, (4R)-

Biological Activity

[Description]:

BET-BAY 002 is a potent BET inhibitor; shows efficacy in a multiple myeloma model.

[Related Catalog]:

Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain
Research Areas >> Cancer

[Related Small Molecules]

(+)-JQ1 | GSK126 | Tazemetostat (EPZ-6438) | Birabresib (OTX015) | A 485 | Curcumin | ARV-771 | ARV-825 | I-BET762 | BI 2536 | GSK343 | C646 | 3-Deazaneplanocin A (hydrochloride) | I-BET151 | 666-15

Chemical & Physical Properties

[ Density]:
1.4±0.1 g/cm3

[ Boiling Point ]:
635.7±65.0 °C at 760 mmHg

[ Molecular Formula ]:
C22H18ClN5O

[ Molecular Weight ]:
403.864

[ Flash Point ]:
338.3±34.3 °C

[ Exact Mass ]:
403.119995

[ LogP ]:
3.92

[ Vapour Pressure ]:
0.0±1.9 mmHg at 25°C

[ Index of Refraction ]:
1.715

[ Storage condition ]:
2-8℃

Related Compounds