c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm

Names

[ CAS No. ]:
1647119-71-8

[ Name ]:
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm

Biological Activity

[Description]:

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm is a is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.25 and 0.05 nM for hV2R and rV2R, respectively[1].

[Related Catalog]:

Signaling Pathways >> Others >> Others
Research Areas >> Neurological Disease

[Target]

EC50: 0.25 nM (hV2R), 0.05 nM (rV2R)[1]


[References]

[1]. Wiśniewski K, et al. Discovery of Potent, Selective, and Short-Acting Peptidic V2 Receptor Agonists. J Med Chem. 2019 May 23;62(10):4991-5005.

Chemical & Physical Properties

[ Molecular Formula ]:
C47H69ClN12O9S2

[ Molecular Weight ]:
1045.71

Related Compounds