H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-Lys-tBu-Gly-Cys-2-Nal-NH2 trifluoroacetate salt (Disulfide bond)
Names
[ CAS No. ]:
209006-18-8
[ Name ]:
H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-Lys-tBu-Gly-Cys-2-Nal-NH2 trifluoroacetate salt (Disulfide bond)
[Synonym ]:
prl-2915
Biological Activity
[Description]:
[Related Catalog]:
[Target]
hsst2:12 nM (Ki)
hsst3:100 nM (Ki)
hsst5:520 nM (Ki)
hsst4:895 nM (Ki)
hsst1:>1000 nM (Ki)
hsst2:1.8 nM (IC50, rat antagonist bioassay versus somatostatin)
rat urotensin II receptor:293 nM (Ki)
human urotensin II receptor:562 nM (Ki)
[In Vitro]
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C59H71ClN12O8S2
[ Molecular Weight ]:
1175.85
[ Exact Mass ]:
1174.46000
[ PSA ]:
378.11000
[ LogP ]:
7.94310