L-797591

Names

[ CAS No. ]:
217480-24-5

[ Name ]:
L-797591

Biological Activity

[Description]:

L-797591 is a selective somatostatin receptor subtype 1 (SSTR1) agonist[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Somatostatin Receptor
Research Areas >> Metabolic Disease

[In Vitro]

L-797591 (10 nM; 1 h) 减少 GLP-1 诱导的 RINm5F 细胞的胰岛素分泌[1]。

[References]

[1]. Stark A, et al. Somatostatin inhibits glucagon-like peptide-1-induced insulin secretion and proliferation of RINm5F insulinoma cells. Regul Pept. 2002 Oct 15;108(2-3):97-102.  

Chemical & Physical Properties

[ Molecular Formula ]:
C38H49N5O2

[ Molecular Weight ]:
607.83


Related Compounds