PROTAC ERRα Degrader-1

Names

[ Name ]:
PROTAC ERRα Degrader-1

Biological Activity

[Description]:

PROTAC ERRalpha Degrader-1 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRalpha Degrader-1 is an estrogen-related receptor alpha (ERRa) degrader[1].

[Related Catalog]:

Signaling Pathways >> Others >> Estrogen Receptor/ERR

Research Areas >> Cancer

Signaling Pathways >> PROTAC >> PROTAC

[References]

[1]. Peng L, et al. Identification of New Small-Molecule Inducers of Estrogen-related Receptor α (ERRα) Degradation. ACS Med Chem Lett. 2019 Apr 12;10(5):767-772.

Chemical & Physical Properties

[ Molecular Formula ]:
C₅₄H₄₉Cl₂F₆N₇O₈

[ Molecular Weight ]:
1108.91

[ Storage condition ]:
2-8°C