BET bromodomain inhibitor 2

Names

[ CAS No. ]:
2414195-69-8

[ Name ]:
BET bromodomain inhibitor 2

Biological Activity

[Description]:

BET bromodomain inhibitor 2 is a potent BET bromodomain inhibitor with an IC50 of 14.1 µM[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[References]

[1]. J P Hilton-Proctor, et al. Substituted 1-methyl-4-phenylpyrrolidin-2-ones - Fragment-based design of N-methylpyrrolidone-derived bromodomain inhibitors. Eur J Med Chem. 2020 Apr 1;191:112120.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₃H₃₀N₂O₅S

[ Molecular Weight ]:
446.56

Related Compounds