(R)-VT104

Names

[ Name ]:
(R)-VT104

Biological Activity

[Description]:

(R)-VT104 is the R-enantiomer of VT104. (R)-VT104 shows an IC50 value of 0.1-1 μΜ for firefly luciferase. VT104 is an orally active and pan-TEAD auto-palmitoylation inhibitor[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Stem Cell/Wnt >> YAP

[References]

[1]. Konradi, Andrei W, et al. Preparation of substituted naphthalene-2-carboxamide derivatives useful for treatment of cancer. WO2020097389.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₅H₁₉F₃N₂O

[ Molecular Weight ]:
420.43

(R)-VT104

Names

Biological Activity

Chemical & Physical Properties

Related Compounds