<Suppliers Price>

PCSK9-IN-12

Names

[ CAS No. ]:
2455427-91-3

[ Name ]:
PCSK9-IN-12

Biological Activity

[Description]:

PCSK9-IN-12 is a heteroaryl compound. PCSK9-IN-12 has bind affinity for PCSK9 with a Kd value of ＜200 nM. PCSK9-IN-12 can be used for the research of cholesterol metabolism[1].

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Ser/Thr Protease
Research Areas >> Metabolic Disease

[In Vitro]

PCSK9-IN-12 (compound 458B) 对 PCSK9 具有亲和力，Kd 值为 <200 nM[1]。

[References]

[1]. Michael H. Serrano-Wu, et al. Pcsk9 inhibitors and methods of use thereof. Patent. WO2020150474A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C20H20F2N6O2

[ Molecular Weight ]:
414.41

Related Compounds