μ opioid receptor agonist 2

Names

[ CAS No. ]:
2671755-38-5

[ Name ]:
μ opioid receptor agonist 2

Biological Activity

[Description]:

μ opioid receptor agonist 2 (Compound H-3)is an optically pure oxaspiro ring substituted pyrrolopyrazole derivative, acts as a MOR receptor agonist and can be used for the research of pain and pain related diseases[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Opioid Receptor
Signaling Pathways >> Neuronal Signaling >> Opioid Receptor
Research Areas >> Neurological Disease

[Target]

EC50: 17 nM (cAMP)[1]


[References]

[1]. Azabicyclic substituted oxaspiro derivative, preparation method therefor and medical use thereof. WO2021143801A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C25H34N4O

[ Molecular Weight ]:
406.56


Related Compounds