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BRD4-BD1/2-IN-2

Names

[ CAS No. ]:
2743464-27-7

[ Name ]:
BRD4-BD1/2-IN-2

Biological Activity

[Description]:

BRD4-BD1/2-IN-2 is a potent BRD4 BD2 inhibitor with IC50s of <0.5 nM and <300 nM for BRD4 BD2 and BRD4 BD1, respectively (WO2021233371A1, compound 2)[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[References]

[1]. Compound functioning as bromodomain protein inhibitor, and composition. WO2021233371A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C30H33N5O4

[ Molecular Weight ]:
527.61


Related Compounds