DC-BPi-03

Names

[ CAS No. ]:
2758411-46-8

[ Name ]:
DC-BPi-03

Biological Activity

[Description]:

DC-BPi-03 is a potent BPTF-BRD inhibitor with an IC50 of 698.3 nM and a Kd of 2.81 μM[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[References]

[1]. Tian Lu, et al. Discovery of High-Affinity Inhibitors of the BPTF Bromodomain. J Med Chem. 2021 Aug 26;64(16):12075-12088.  

Chemical & Physical Properties

[ Molecular Formula ]:
C14H14N4O2S

[ Molecular Weight ]:
302.35

Related Compounds