BRD4-BD1-IN-1

Names

[ CAS No. ]:
2761321-18-8

[ Name ]:
BRD4-BD1-IN-1

Biological Activity

[Description]:

BRD4-BD1-IN-1 (Compound 9a) is a BRD4-BD1 inhibitor with an IC50 of 38.20 μM[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[Target]

BRD4 BD1:38.20 μM (IC50)

[References]

[1]. Chang Y, et al. Design, synthesis, biological evaluation, and molecular docking of 1, 7-dibenzyl-substituted theophylline derivatives as novel BRD4-BD1-selective inhibitors. Medicinal Chemistry Research, 2021, 30(8): 1453-1468.

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₆H₁₅BrN₄O₄

[ Molecular Weight ]:
407.22

Related Compounds