d[Cha4]-AVP TFA

Names

[ Name ]:
d[Cha4]-AVP TFA

[Synonym ]:
3-Mercaptopropionyl-Tyr-Phe-b-cyclohexyl-Ala-Asn-Cys-Pro-Arg-Gly-NH2

Biological Activity

[Description]:

d[Cha4]-AVP is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). d[Cha4]-AVP stimulates ACTH and corticosterone secretion and exhibits negligible vasopressor activity in vivo.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Vasopressin Receptor

Chemical & Physical Properties

[ Molecular Formula ]:
C₅₀H₇₁N₁₃O₁₁S₂

[ Molecular Weight ]:
1096.33000

[ Exact Mass ]:
1095.50000

[ PSA ]:
469.92000

[ LogP ]:
3.30320

Safety Information

[ Hazard Codes ]:
Xi

d[Cha4]-AVP TFA

Names

Biological Activity

Chemical & Physical Properties

Safety Information

Related Compounds