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Taranabant (1R,2R) stereoisomer

Names

[ CAS No. ]:
701977-08-4

[ Name ]:
Taranabant (1R,2R) stereoisomer

[Synonym ]:
Propanamide, N-[(1R,2R)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-methyl-2-[[5-(trifluoromethyl)-2-pyridinyl]oxy]-
N-[(2R,3R)-4-(4-Chlorophenyl)-3-(3-cyanophenyl)-2-butanyl]-2-methyl-2-{[5-(trifluoromethyl)-2-pyridinyl]oxy}propanamide

Biological Activity

[Description]:

Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Cannabinoid Receptor
Research Areas >> Others

[References]

[1]. William K. Hagmann, et al. Substituted amides active at the cannabinoid-1 receptor. WO 2004048317 A1.


[Related Small Molecules]

WIN 55212-2 mesylate | AM251 | Taranabant | SR144528 | Bay 59-3074 | Org 27569 | Otenabant | GW842166X | A-836339 | BML-190 | JD-5037 | (±)-SLV319 | Pregnenolone | Anandamide | 2-arachidonoylglycerol

Chemical & Physical Properties

[ Density]:
1.3±0.1 g/cm3

[ Boiling Point ]:
634.2±55.0 °C at 760 mmHg

[ Molecular Formula ]:
C27H25ClF3N3O2

[ Molecular Weight ]:
515.955

[ Flash Point ]:
337.4±31.5 °C

[ Exact Mass ]:
515.158752

[ LogP ]:
7.13

[ Vapour Pressure ]:
0.0±1.9 mmHg at 25°C

[ Index of Refraction ]:
1.575

Related Compounds