<Suppliers Price>

Sarmazenil

Names

[ CAS No. ]:
78771-13-8

[ Name ]:
Sarmazenil

[Synonym ]:
Sarmazenilum
Sarmazenil
sarmazenil[inn]
ethyl 7-chloro-5-methyl-6-oxo-5,6-dihydro-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate
Sarmazenilum [INN-Latin]
ethyl 7-chloro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate

Biological Activity

[Description]:

Sarmazenil is a benzodiazepine receptor antagonist.

[Related Catalog]:

Signaling Pathways >> Membrane Transporter/Ion Channel >> GABA Receptor
Signaling Pathways >> Neuronal Signaling >> GABA Receptor
Research Areas >> Neurological Disease

[Target]

Benzodiazepine receptor[1]


[References]

[1]. Gath I, et al. Electrophysiological aspects of benzodiazepine antagonists, Ro 15-1788 and Ro 15-3505. Br J Clin Pharmacol. 1984 Oct;18(4):541-7.


[Related Small Molecules]

(+)-Bicuculline | Picrotoxin | Aminooxyacetic acid hemihydrochloride | Riluzole | Baclofen | basmisanil | (R)-Baclofen | Etifoxine | Etomidate | Ginkgolide A | NS-11394 | 5alpha-Pregnan-3alpha-ol-20-one | CGP 52432 | L-655,708 | SAGE-217

Chemical & Physical Properties

[ Density]:
1.43g/cm3

[ Boiling Point ]:
554ºC at 760 mmHg

[ Molecular Formula ]:
C15H14ClN3O3

[ Molecular Weight ]:
319.74300

[ Flash Point ]:
288.9ºC

[ Exact Mass ]:
319.07200

[ PSA ]:
64.43000

[ LogP ]:
2.22590

[ Index of Refraction ]:
1.658

[ Storage condition ]:
2-8℃

Synthetic Route

Click to get detail synthetic route

Precursor & DownStream

Precursor

DownStream

Related Compounds