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Histone Acetyltransferase Inhibitor II

Names

[ CAS No. ]:
932749-62-7

[ Name ]:
Histone Acetyltransferase Inhibitor II

[Synonym ]:
HistoneAcetyltransferaseInhibitorII
Histone Acetyltransferase Inhibitor II

Biological Activity

[Description]:

Histone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 µM; Histone Acetyltransferase Inhibitor II can be used in cancer research.

[Related Catalog]:

Signaling Pathways >> Epigenetics >> Histone Acetyltransferase
Research Areas >> Cancer

[Target]

IC50：5 µM (p300)[1]


[In Vitro]

Histone Acetyltransferase Inhibitor II 是一种有效的，细胞渗透的 p300 抑制剂，IC50 值为 5 µM，可用于癌症研究。

[References]

[1]. Costi R, et al. Cinnamoyl compounds as simple molecules that inhibit p300 histone acetyltransferase. J Med Chem. 2007 Apr 19;50(8):1973-7. Epub 2007 Mar 10.


[Related Small Molecules]

A 485 | Curcumin | C646 | CPI-637 | SGC-CBP30 | GNE-272 | MG149 | WM 1119 | anacardic acid | I-CBP 112 | MOZ-IN-3 | PF-CBP1 hydrochloride | Remodelin hydrobromide | TPOP146 | GNE-781

Chemical & Physical Properties

[ Molecular Formula ]:
C20H16Br2O3

[ Molecular Weight ]:
464.14700

[ Exact Mass ]:
461.94700

[ PSA ]:
57.53000

[ LogP ]:
5.84280

[ Storage condition ]:
2-8℃

Related Compounds