CBP/p300-IN-14

Names

[ CAS No. ]:
2725036-10-0

[ Name ]:
CBP/p300-IN-14

Biological Activity

[Description]:

CBP/p300-IN-14 is a potent inhibitor of CBP/EP300 (lysine acetyltransferase) with an IC50 of 3.3 nM (extracted from patent WO2021213521A1, compound 27)[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Histone Acetyltransferase
Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[Target]

3.3 nM (CBP/EP300)[1]


[References]

[1]. Wang, Lisha, et al. Cbp/ep300 inhibitor and use thereof. Patent WO2021213521A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C30H31F2N7O2

[ Molecular Weight ]:
559.61

Related Compounds