BRD4 Inhibitor-19

Names

[ CAS No. ]:
2757865-63-5

[ Name ]:
BRD4 Inhibitor-19

Biological Activity

[Description]:

BRD4 Inhibitor-19 is a BET inhibitor with an IC50 of 55 nM for BRD4-BD1. BRD4 Inhibitor-19 can be used for multiple myeloma research[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[Target]

BD1:55 nM (IC50)

[References]

[1]. Lincheng Fang, et al. Discovery of 3,5-dimethylisoxazole derivatives as novel, potent inhibitors for bromodomain and extraterminal domain (BET) family. Bioorg Med Chem. 2021 Jun 1;39:116133.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₉H₂₅N₅O₃

[ Molecular Weight ]:
491.54

Related Compounds