P2X7 receptor antagonist-3
Names
[ CAS No. ]:
1627900-92-8
[ Name ]:
P2X7 receptor antagonist-3
Biological Activity
[Description]:
P2X7 receptor antagonist-3 is a potent P2X7 receptor antagonist with P2X7R IC50 values of 4.2 nM in humans and 6.8 nM in rats[1].
[Related Catalog]:
[Target]
hP2X7R:4.2 nM (IC50)
rP2X7R:6.8 nM (IC50)
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C17H12ClF3N6O
[ Molecular Weight ]:
408.76