AKT-IN-12
Names
[ CAS No. ]:
2396718-52-6
[ Name ]:
AKT-IN-12
Biological Activity
[Description]:
AKT-IN-12 (compound 3e) is a potent Akt kinase inhibitor with an IC50 value of 0.55 μM. AKT-IN-12 induces G0/G1 cell cycle arrest and apoptosis. AKT-IN-12 also inhibits p-AKT, p-ERK, and activates p-JNK, JNK. AKT-IN-12 can be used for researching leukemia[1].
[Related Catalog]:
[Target]
IC50: 0.55 μM (Akt)[1]
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C42H46N2O7S
[ Molecular Weight ]:
722.89