Glyoxalase I inhibitor 5

Names

[ CAS No. ]:
2455508-17-3

[ Name ]:
Glyoxalase I inhibitor 5

Biological Activity

[Description]:

Glyoxalase I inhibitor 5 (Compound 9h) is a glyoxalase I (Glo-I) inhibitor with an IC50 of 1.28 μM. Glyoxalase I inhibitor 5 can be used as anticancer agent[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Others >> Others

[Target]

IC50: 1.28 μM (Glo-I)[1]


[References]

[1]. Al-Oudat BA, et al. Design, synthesis and biological evaluation of novel glyoxalase I inhibitors possessing diazenylbenzenesulfonamide moiety as potential anticancer agents. Bioorg Med Chem. 2020 Aug 15;28(16):115608.

Chemical & Physical Properties

[ Molecular Formula ]:
C16H14N4O3S

[ Molecular Weight ]:
342.37

Related Compounds