PAL-4

Names

[ CAS No. ]:
2609594-35-4

[ Name ]:
PAL-4

Biological Activity

[Description]:

PAL-4 (compound 4) is a potent, selective and reversible Lysophospholipase-like 1 (LYPLAL1) activator with EC50 value of 0.39 μM and 0.49 μM for mice LYPLAL1 and huamn LYPLAL1, respectively. PAL-4 can be used for researching metabolic disorders[1].

[Related Catalog]:

Signaling Pathways >> Others >> Others
Research Areas >> Metabolic Disease

[Target]

IC50: 0.39 μM (mice LYPLAL1), 0.49 μM (human LYPLAL1)[1]


[References]

[1]. Kok BP, et al. Discovery of small-molecule enzyme activators by activity-based protein profiling. Nat Chem Biol. 2020;16(9):997-1005.

Chemical & Physical Properties

[ Molecular Formula ]:
C17H15ClN4O3S2

[ Molecular Weight ]:
422.91


Related Compounds