vMIP-II (1-21)
Names
[ CAS No. ]:
265650-93-9
[ Name ]:
vMIP-II (1-21)
Biological Activity
[Description]:
vMIP-II (1-21) is a CXCR4 antagonist. vMIP-II has broad-spectrum interaction with CC and CXC chemokine receptors. vMIP-II (1-21) binds with CXCR4 with an IC50 value of 190 nM for competing with CXCR4 binding of 125I-SDF-1R[1].
[Related Catalog]:
[In Vitro]
vMIP-II (1-21) (0.01-10 μM) 可与趋化因子受体 CXCR4 结合[1]。 vMIP-II (1-21) (25-200 μM) 抑制 CXCR4 介导 T 和双亲性 HIV-1 gp120 介导的细胞-细胞融合[1]。 vMIP-II (1-21) (100 μM) 剂量依赖性地抑制的趋化活性[1]。
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C108H169N33O27S
[ Molecular Weight ]:
2425.84