Androgen receptor antagonist 3

Names

[ CAS No. ]:
353484-46-5

[ Name ]:
Androgen receptor antagonist 3

Biological Activity

[Description]:

Androgen receptor antagonist 3 (Compound C18) is an androgen receptor (AR) antagonist with an IC50 of 2.4 μM. Androgen receptor antagonist 3 shows anticancer activities[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Others >> Androgen Receptor

[Target]

IC50: 2.4 μM (Androgen receptor)[1]


[References]

[1]. Tang Q, et al. Novel androgen receptor antagonist identified by structure-based virtual screening, structural optimization, and biological evaluation. Eur J Med Chem. 2020 Apr 15;192:112156.

Chemical & Physical Properties

[ Molecular Formula ]:
C22H18ClN

[ Molecular Weight ]:
331.84

Related Compounds