Mergetpa

Names

[ Name ]:
Mergetpa

[Synonym ]:
dl-2-mercaptomethyl-3-guanidinoethylthiopropanoic acid

Biological Activity

[Description]:

Mergetpa is a carboxypeptidase inhibitor used to block the conversion of kinins and B2 receptor antagonists to metabolites lacking the C-terminal arginine[1].

[Related Catalog]:

Research Areas >> Others

Signaling Pathways >> Metabolic Enzyme/Protease >> Carboxypeptidase

[References]

[1]. D Regoli, et al. Conversion of kinins and their antagonists into B1 receptor activators and blockers in isolated vessels. Eur J Pharmacol. 1986 Aug 15;127(3):219-24.

Chemical & Physical Properties

[ Molecular Formula ]:
C₇H₁₅N₃O₂S₂

[ Molecular Weight ]:
237.34

[ Exact Mass ]:
237.06100

[ PSA ]:
163.30000

[ LogP ]:
1.02420

Safety Information

[ HS Code ]:
2930909090

Customs

[ HS Code ]: 2930909090

[ Summary ]:
2930909090. other organo-sulphur compounds. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:30.0%