1356013-39-2
1356013-39-2 structure
- Name: TAK1-IN-1
- Chemical Name: TAK1-IN-1
- CAS Number: 1356013-39-2
- Molecular Formula: C17H12N4O2S
- Molecular Weight: 336.369
- Create Date: 2020-01-11 19:10:49
- Modify Date: 2023-02-19 17:30:46
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TAK1-IN-1 is a potent, selective, Type I (ATP-competitive, DFG-in) TAK1 inhibitor with Kd of 59 nM, a thienopyrimidine scaffold that serves as a good starting point for medicinal chemistry.
| Name | TAK1-IN-1 |
|---|
| Description | TAK1-IN-1 is a potent, selective, Type I (ATP-competitive, DFG-in) TAK1 inhibitor with Kd of 59 nM, a thienopyrimidine scaffold that serves as a good starting point for medicinal chemistry. |
|---|---|
| References | References 1. Miura T, et al. Bioorg Med Chem Lett. 2017 Feb 15;27(4):1031-1036. View Related Products by Target TAK1 |
| Molecular Formula | C17H12N4O2S |
|---|---|
| Molecular Weight | 336.369 |