371131-16-7
371131-16-7 structure
- Name: PZ-128
- Chemical Name: IYT6MP4NS9
- CAS Number: 371131-16-7
- Molecular Formula: C55H99N13O9
- Molecular Weight: 1086.456
- Create Date: 2021-01-09 18:19:06
- Modify Date: 2024-04-12 20:35:46
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PZ-128 (P1pal-7), a cell-penetrating lipopeptide pepducin, is a first-in-class, specific and reversible protease-activated receptor-1 (PAR1) antagonist. PZ-128 targets the cytoplasmic surface of PAR1 and interrupts signaling to internally-located G (PAR1-G) proteins. PZ-128 has antiplatelet, anti-metastatic, anti-angiogenic and anticancer effects.
| Name | IYT6MP4NS9 |
|---|---|
| Synonyms |
IYT6MP4NS9
N2-Palmitoyl-L-lysyl-L-lysyl-L-seryl-L-arginyl-L-alanyl-L-leucyl-L-phenylalaninamide L-Phenylalaninamide, N2-(1-oxohexadecyl)-L-lysyl-L-lysyl-L-seryl-L-arginyl-L-alanyl-L-leucyl- |
| Density | 1.2±0.1 g/cm3 |
|---|---|
| Molecular Formula | C55H99N13O9 |
| Molecular Weight | 1086.456 |
| Exact Mass | 1085.768921 |
| LogP | 4.95 |
| Index of Refraction | 1.585 |
| Storage condition | -20°C |