2535970-65-9
2535970-65-9 structure
- Name: EST73502 hydrochloride
- Chemical Name: EST73502 hydrochloride
- CAS Number: 2535970-65-9
- Molecular Formula: C19H27ClF2N2O2
- Molecular Weight: 388.88
- Create Date: 2021-09-11 19:50:30
- Modify Date: 2024-01-05 17:16:56
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EST73502 hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 hydrochloride has antinociceptive activity.
| Name | EST73502 hydrochloride |
|---|
| Description | EST73502 hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 hydrochloride has antinociceptive activity. |
|---|
| Molecular Formula | C19H27ClF2N2O2 |
|---|---|
| Molecular Weight | 388.88 |