Shanghai Nianxing Industrial Co., Ltd
China
Product Name: KSK94
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Purity: 99.56%
Stocking Period: 10 Day
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2566716-07-0

2566716-07-0 structure

2566716-07-0 structure

Name: KSK94
Chemical Name: KSK94
CAS Number: 2566716-07-0
Molecular Formula: C₂₅H₂₆N₄O
Molecular Weight: 398.50
Catalog: Signaling Pathways GPCR/G Protein Histamine Receptor
Create Date: 2023-09-19 16:36:08
Modify Date: 2024-01-12 19:41:39
KSK94 is a high-affinity histamine H3 receptor antagonist, with Kis of 7.9, 2958, 75.2 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK94 can be used for research of nociceptive and neuropathic pain[1].

Name	KSK94

Description	KSK94 is a high-affinity histamine H3 receptor antagonist, with Kis of 7.9, 2958, 75.2 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK94 can be used for research of nociceptive and neuropathic pain[1].
Related Catalog	Signaling Pathways >> Immunology/Inflammation >> Histamine Receptor Research Areas >> Neurological Disease Signaling Pathways >> GPCR/G Protein >> Sigma Receptor Signaling Pathways >> GPCR/G Protein >> Histamine Receptor
Target	7.9, 2958, 75.2 nM (H3 receptor, sigma-1, sigma-2 receptor)[1]
References	[1]. Szczepańska K, et al. Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain. J Med Chem. 2023 Jul 27;66(14):9658-9683.

Molecular Formula	C₂₅H₂₆N₄O
Molecular Weight	398.50