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1260075-17-9

1260075-17-9 structure
1260075-17-9 structure
  • Name: Mitapivat
  • Chemical Name: N-(4-(4-(cyclopropylmethyl)piperazine-1-carbonyl)phenyl)quinoline-8-sulfonamide
  • CAS Number: 1260075-17-9
  • Molecular Formula: C24H26N4O3S
  • Molecular Weight: 450.55300
  • Catalog: Research Areas Cancer
  • Create Date: 2017-05-13 15:36:31
  • Modify Date: 2024-01-03 20:08:39
  • Mitapivat is a potent human R-type pyruvate kinase (PKR) inhibitor; also shows potency for mutant PKR including R510Q PKR, R532W PKR, T384W PKR etc.

Name N-(4-(4-(cyclopropylmethyl)piperazine-1-carbonyl)phenyl)quinoline-8-sulfonamide
Synonyms PKM2 activator 1020
Mitapivat
Description Mitapivat is a potent human R-type pyruvate kinase (PKR) inhibitor; also shows potency for mutant PKR including R510Q PKR, R532W PKR, T384W PKR etc.
Related Catalog
References

[1]. PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY. Patent WO/2012/151451A1

Molecular Formula C24H26N4O3S
Molecular Weight 450.55300
Exact Mass 450.17300
PSA 90.99000
LogP 4.23300