Name | N-(4-(4-(cyclopropylmethyl)piperazine-1-carbonyl)phenyl)quinoline-8-sulfonamide |
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Synonyms |
PKM2 activator 1020
Mitapivat |
Description | Mitapivat is a potent human R-type pyruvate kinase (PKR) inhibitor; also shows potency for mutant PKR including R510Q PKR, R532W PKR, T384W PKR etc. |
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Related Catalog | |
References |
[1]. PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY. Patent WO/2012/151451A1 |
Molecular Formula | C24H26N4O3S |
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Molecular Weight | 450.55300 |
Exact Mass | 450.17300 |
PSA | 90.99000 |
LogP | 4.23300 |