607742-80-3

607742-80-3 structure

Name: GSK215083
Chemical Name: 4-(3-fluorophenyl)sulfonyl-8-(4-methylpiperazin-1-yl)quinoline
CAS Number: 607742-80-3
Molecular Formula: C₂₀H₂₀FN₃O₂S
Molecular Weight: 385.46
Create Date: 2017-07-18 14:56:54
Modify Date: 2024-01-10 04:50:12
GSK215083 is a high affinity 5-HT6 receptor antagonist. GSK215083 can serves as a promising 5-HT6 radioligand candidate by radiolabeled with (11)C via methylation[1].

Name	4-(3-fluorophenyl)sulfonyl-8-(4-methylpiperazin-1-yl)quinoline
Synonyms	unii-8gfe8j4n0z

Description	GSK215083 is a high affinity 5-HT6 receptor antagonist. GSK215083 can serves as a promising 5-HT6 radioligand candidate by radiolabeled with (11)C via methylation[1].
Related Catalog	Research Areas >> Others Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor
Target	5-HT6 Receptor
References	[1]. Parker CA, et al. Radiosynthesis and characterization of 11C-GSK215083 as a PET radioligand for the 5-HT6 receptor. J Nucl Med. 2012 Feb;53(2):295-303.