Acetyl-Calpastatin (184-210) (human) trifluoroacetate salt
Modify Date: 2024-01-19 15:44:42
Acetyl-Calpastatin (184-210) (human) trifluoroacetate salt structure
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Common Name | Acetyl-Calpastatin (184-210) (human) trifluoroacetate salt | ||
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| CAS Number | 123714-50-1 | Molecular Weight | 3177.63000 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C142H230N36O44S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Acetyl-Calpastatin (184-210) (human) trifluoroacetate saltAcetyl-Calpastatin(184-210)(human) is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin L, respectively[1][2]. |
| Name | Acetyl-Calpastatin (184-210) (human) |
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| Description | Acetyl-Calpastatin(184-210)(human) is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin L, respectively[1][2]. |
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| Related Catalog | |
| In Vitro | Acetyl-Calpastatin(184-210)(human) (peptide 1; 12.5-100 μM) inhibits calpains in LCLC 103H cells with an IC50 of 27 μM[1]. |
| References |
[1]. Ferdinando Fiorino, et al. A new cell-permeable calpain inhibitor. J Pept Sci. 2007 Jan;13(1):70-3. |
| Molecular Formula | C142H230N36O44S |
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| Molecular Weight | 3177.63000 |
| Exact Mass | 3175.66000 |
| PSA | 1311.44000 |
| LogP | 3.43000 |
| Appearance of Characters | powder |
| Storage condition | −20°C |
| Water Solubility | H2O: 1 mg/mL |
| WGK Germany | 3 |
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