Cav 3.2 inhibitor 4

Modify Date: 2024-09-18 09:40:10

Cav 3.2 inhibitor 4 Structure
Cav 3.2 inhibitor 4 structure
Common Name Cav 3.2 inhibitor 4
CAS Number 1416984-93-4 Molecular Weight 459.41
Density N/A Boiling Point N/A
Molecular Formula C21H32Cl2N4O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Cav 3.2 inhibitor 4


Cav 3.2 inhibitor 4 (compound 21) is a potent, peripherally restricted, selective T-type calcium channel (Cav3.2) inhibitor, with an IC50 of 0.6 μM. Cav 3.2 inhibitor 4 can be used for the research of atrial fibrillation[1].

 Names

Name Cav 3.2 inhibitor 4

 Cav 3.2 inhibitor 4 Biological Activity

Description Cav 3.2 inhibitor 4 (compound 21) is a potent, peripherally restricted, selective T-type calcium channel (Cav3.2) inhibitor, with an IC50 of 0.6 μM. Cav 3.2 inhibitor 4 can be used for the research of atrial fibrillation[1].
Related Catalog
References

[1]. Giordanetto F, et, al. Discovery of N-[[1-[2-(tert-butylcarbamoylamino)ethyl]-4-(hydroxymethyl)-4-piperidyl]methyl]-3,5-dichloro-benzamide as a selective T-type calcium channel (Cav3.2) inhibitor. Bioorg Med Chem Lett. 2013 Jan 1;23(1):119-24.  

 Chemical & Physical Properties

Molecular Formula C21H32Cl2N4O3
Molecular Weight 459.41