c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2

Modify Date: 2024-01-09 19:01:33

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 Structure
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 structure
Common Name c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
CAS Number 1647119-61-6 Molecular Weight 946.58
Density N/A Boiling Point N/A
Molecular Formula C42H60ClN11O8S2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2


c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively[1].

 Names

Name c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2

  Biological Activity

Description c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively[1].
Related Catalog
Target

EC50: 0.07 nM (hV2R), 0.02 nM (rV2R)[1]

References

[1]. Wiśniewski K, et al. Discovery of Potent, Selective, and Short-Acting Peptidic V2 Receptor Agonists. J Med Chem. 2019 May 23;62(10):4991-5005.

 Chemical & Physical Properties

Molecular Formula C42H60ClN11O8S2
Molecular Weight 946.58