KRpep-2d structure
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Common Name | KRpep-2d | ||
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CAS Number | 2098181-84-9 | Molecular Weight | 2560.02 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C109H183N43O25S2 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of KRpep-2dKRpep-2d is a potent K-Ras inhibitor and inhibits proliferation of K-Ras-driven cancer cells. KRpep-2d can be used for cancer research[1]. |
Name | KRpep-2d |
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Description | KRpep-2d is a potent K-Ras inhibitor and inhibits proliferation of K-Ras-driven cancer cells. KRpep-2d can be used for cancer research[1]. |
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Related Catalog | |
Target |
K-RAS |
In Vitro | KRpep-2d has cyclic structure with importance for K-Ras inhibitory activity. Leu77 , Ile9 and Asp12 are critical amino acid residues for the K-Ras inhibitory activity of KRpep-2d[1]. KRpep-2d (10-30 μM) has inhibitory activity of A427 cells with the proliferation rates of 68.3% (10 μM) and 48.3% (10 μM)[1]. |
References |
Molecular Formula | C109H183N43O25S2 |
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Molecular Weight | 2560.02 |