BCX 1470 (methanesulfonate) structure
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Common Name | BCX 1470 (methanesulfonate) | ||
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CAS Number | 217099-44-0 | Molecular Weight | 398.47700 | |
Density | N/A | Boiling Point | 509.9ºC at 760 mmHg | |
Molecular Formula | C15H14N2O5S3 | Melting Point | N/A | |
MSDS | N/A | Flash Point | 262.2ºC |
Use of BCX 1470 (methanesulfonate)BCX 1470 inhibits the esterolytic activity of factor D (IC50=96 nM) and C1s (IC50=1.6 nM), 3.4- and 200-fold better, respectively, than that of trypsin.IC50 Value: 96 nM (Factor D); 1.6 nM (C1s); 326 nM (Trypsin) [1]Target: Factor D; C1sBCX 1470(Thrombin inhibitor) is serine protease inhibitor.BCX 1470(Thrombin inhibitor) blocks the esterolytic and hemolytic activities of the complement enzymes Cls and factor D in vitro, also blocked development of RPA-induced edema in the rat. |
Name | 2-Thiophenecarboxylic acid 2-(aminoiminomethyl)benzo[b]thiophen-6-yl ester methanesulfonate (1:1) |
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Synonym | More Synonyms |
Description | BCX 1470 inhibits the esterolytic activity of factor D (IC50=96 nM) and C1s (IC50=1.6 nM), 3.4- and 200-fold better, respectively, than that of trypsin.IC50 Value: 96 nM (Factor D); 1.6 nM (C1s); 326 nM (Trypsin) [1]Target: Factor D; C1sBCX 1470(Thrombin inhibitor) is serine protease inhibitor.BCX 1470(Thrombin inhibitor) blocks the esterolytic and hemolytic activities of the complement enzymes Cls and factor D in vitro, also blocked development of RPA-induced edema in the rat. |
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Related Catalog | |
References |
Boiling Point | 509.9ºC at 760 mmHg |
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Molecular Formula | C15H14N2O5S3 |
Molecular Weight | 398.47700 |
Flash Point | 262.2ºC |
Exact Mass | 398.00600 |
PSA | 195.40000 |
LogP | 4.85090 |
Storage condition | 2-8℃ |
BCX 1470 methanesulfonate |
BCX 1470 (methanesulfonate) |