KDM4-IN-4 structure
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Common Name | KDM4-IN-4 | ||
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CAS Number | 2230475-63-3 | Molecular Weight | 245.36 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C16H23NO | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of KDM4-IN-4KDM4-IN-4 (compound 47) is a potent histone lysine demethylase 4 (KDM4) inhibitor with a modest affinity binding to ~80 μM for KDM4A-Tudor domain. KDM4-IN-4 can inhibit H3K4Me3 binding to the Tudor domain in cells with an EC50 value of 105 μM. KDM4-IN-4 can be used for researching anticancer[1]. |
Name | KDM4-IN-4 |
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Description | KDM4-IN-4 (compound 47) is a potent histone lysine demethylase 4 (KDM4) inhibitor with a modest affinity binding to ~80 μM for KDM4A-Tudor domain. KDM4-IN-4 can inhibit H3K4Me3 binding to the Tudor domain in cells with an EC50 value of 105 μM. KDM4-IN-4 can be used for researching anticancer[1]. |
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Related Catalog | |
Target |
KDM4A-Tudor domain:80 μM (Ki) |
References |
Molecular Formula | C16H23NO |
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Molecular Weight | 245.36 |