mGluR2 modulator 1

Modify Date: 2024-01-04 14:37:49

mGluR2 modulator 1 Structure
mGluR2 modulator 1 structure
Common Name mGluR2 modulator 1
CAS Number 2671063-84-4 Molecular Weight 419.40
Density N/A Boiling Point N/A
Molecular Formula C21H20F3N3O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of mGluR2 modulator 1


mGluR2 modulator 1 (compound 95) is a potent and BBB-penetrated mGluR2 (metabotropic glutamate receptor-2) positive allosteric modulator, with an EC50 of 0.03 μM. mGluR2 modulator 1 can be used for psychosis research[1].

 Names

Name mGluR2 modulator 1

 mGluR2 modulator 1 Biological Activity

Description mGluR2 modulator 1 (compound 95) is a potent and BBB-penetrated mGluR2 (metabotropic glutamate receptor-2) positive allosteric modulator, with an EC50 of 0.03 μM. mGluR2 modulator 1 can be used for psychosis research[1].
Related Catalog
Target

mGluR2:0.03 ± 0.0 μM (EC50)

References

[1]. Szabó G, et al. Discovery of dihydropyrazino-benzimidazole derivatives as metabotropic glutamate receptor-2 (mGluR2) positive allosteric modulators (PAMs). Eur J Med Chem. 2020 Jan 15;186:111881.

 Chemical & Physical Properties

Molecular Formula C21H20F3N3O3
Molecular Weight 419.40